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Selective labelling of diazepam-insensitive GABA(A) receptors in vivo using [(3)H]Ro 15-4513

1. Classical benzodiazepines (BZs), such as diazepam, bind to GABA(A) receptors containing α1, α2, α3 or α5 subunits that are therefore described as diazepam-sensitive (DS) receptors. However, the corresponding binding site of GABA(A) receptors containing either an α4 or α6 subunit do not bind the c...

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Autores principales: Pym, Luanda J, Cook, Susan M, Rosahl, Thomas, McKernan, Ruth M, Atack, John R
Formato: Artigo
Lenguaje:Inglês
Publicado: 2005
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC1751217/
https://ncbi.nlm.nih.gov/pubmed/16184188
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0706392
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