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Interactions of metoclopramide and ergotamine with human 5-HT(3A) receptors and human 5-HT reuptake carriers

1. The actions of metoclopramide and ergotamine, drugs which are used as a combined migraine medication, on human (h)5-HT(3A) receptors and 5-HT reuptake carriers, stably expressed in HEK-293 cells, were studied with patch-clamp- and ([(3)H]5-HT)-uptake techniques. 2. At clinical concentrations, met...

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Main Authors: Walkembach, Jan, Brüss, Michael, Urban, Bernd W, Barann, Martin
Formato: Artigo
Idioma:Inglês
Publicado: 2005
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC1751187/
https://ncbi.nlm.nih.gov/pubmed/16041395
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0706351
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