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Affinities of SM-7338 for penicillin-binding proteins and its release from these proteins in Staphylococcus aureus.

SM-7338, a carbapenem antibiotic, had high affinities for penicillin-binding proteins (PBPs) 1, 2, and 4 of Staphylococcus aureus but not for PBP 3 when a competition assay with [14C]benzylpenicillin was used. However, binding of [14C]SM-7338 was saturated for PBP 3 at a concentration of 1 microgram...

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Detalhes bibliográficos
Main Authors: Sumita, Y, Fukasawa, M, Okuda, T
Formato: Artigo
Idioma:Inglês
Publicado em: 1990
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC171622/
https://ncbi.nlm.nih.gov/pubmed/2334163
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