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Serum constituents can affect 2′-& 3′-O-(4-benzoylbenzoyl)-ATP potency at P2X(7) receptors

1. 2′-& 3′-O-(4-benzoylbenzoyl)-ATP (BzATP) is the prototypic agonist for P2X(7) receptors. In this study we demonstrate that bovine serum albumin (BSA) can affect the potency of BzATP at P2X receptors. 2. BzATP potency (pEC(50)) to stimulate ethidium accumulation in cells expressing recombinant...

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Dettagli Bibliografici
Autori principali: Michel, A D, Xing, M, Humphrey, P P A
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2001
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1572703/
https://ncbi.nlm.nih.gov/pubmed/11264244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0703968
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