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Non-competitive pharmacological antagonism at the rabbit B(1) receptor

1. The B(1) receptor for kinins, stimulated by kinin metabolites without the C-terminal Arg residue (e.g., des-Arg(9)-bradykinin (BK) and Lys-des-Arg(9)-BK), is an increasingly recognized molecular target for the development of analgesic and anti-inflammatory drugs. Recently developed antagonists of...

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Autors principals: Larrivée, Jean-François, Gera, Lajos, Houle, Steeve, Bouthillier, Johanne, Bachvarov, Dimcho R, Stewart, John M, Marceau, François
Format: Artigo
Idioma:Inglês
Publicat: 2000
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1572413/
https://ncbi.nlm.nih.gov/pubmed/11053207
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0703656
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