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Direct binding of Cbl to Tyr(568) and Tyr(936) of the stem cell factor receptor/c-Kit is required for ligand-induced ubiquitination, internalization and degradation

The ubiquitin E3 ligase Cbl has been shown to negatively regulate tyrosine kinase receptors, including the stem cell factor receptor/c-Kit. Impaired recruitment of Cbl to c-Kit results in a deregulated positive signalling that eventually can contribute to carcinogenesis. Here, we present results sho...

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Autori principali: Masson, Kristina, Heiss, Elke, Band, Hamid, Rönnstrand, Lars
Natura: Artigo
Lingua:Inglês
Pubblicazione: Portland Press Ltd. 2006
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1570160/
https://ncbi.nlm.nih.gov/pubmed/16780420
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20060464
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