Caricamento...

A771726, the active metabolite of leflunomide, directly inhibits the activity of cyclo-oxygenase-2 in vitro and in vivo in a substrate-sensitive manner

1. The immunosuppressive and anti-inflammatory drug leflunomide has several sites of action, although its precise mode of action is unknown. 2. Here we show in vitro and in vivo that leflunomide and/or its active metabolite A771726, inhibit the activity of cyclo-oxygenase (COX) at doses below those...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Hamilton, Lorna C, Vojnovic, Ivana, Warner, Timothy D
Natura: Artigo
Lingua:Inglês
Pubblicazione: 1999
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1566153/
https://ncbi.nlm.nih.gov/pubmed/10455314
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702708
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !