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Structural insights into substrate traffic and inhibition in acetylcholinesterase

Acetylcholinesterase (AChE) terminates nerve-impulse transmission at cholinergic synapses by rapid hydrolysis of the neurotransmitter, acetylcholine. Substrate traffic in AChE involves at least two binding sites, the catalytic and peripheral anionic sites, which have been suggested to be allosterica...

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Autores principales: Colletier, Jacques-Philippe, Fournier, Didier, Greenblatt, Harry M, Stojan, Jure, Sussman, Joel L, Zaccai, Giuseppe, Silman, Israel, Weik, Martin
Formato: Artigo
Lenguaje:Inglês
Publicado: 2006
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC1500847/
https://ncbi.nlm.nih.gov/pubmed/16763558
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.emboj.7601175
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