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Targeted covalent inactivation of protein kinases by resorcylic acid lactone polyketides

Resorcylic acid lactones containing a cis-enone are susceptible to Michael addition reactions and are potent inhibitors of several protein kinases. A structural-bioinformatics analysis identified a conserved Cys residue in the ATP-binding site of the kinases reported to be inhibited by cis-enone res...

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שמור ב:
מידע ביבליוגרפי
Main Authors: Schirmer, Andreas, Kennedy, Jonathan, Murli, Sumati, Reid, Ralph, Santi, Daniel V.
פורמט: Artigo
שפה:Inglês
יצא לאור: National Academy of Sciences 2006
נושאים:
גישה מקוונת:https://ncbi.nlm.nih.gov/pmc/articles/PMC1449676/
https://ncbi.nlm.nih.gov/pubmed/16537514
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0600445103
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