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Human physiologically based pharmacokinetic model for ACE inhibitors: ramipril and ramiprilat

BACKGROUND: The angiotensin-converting enzyme (ACE) inhibitors have complicated and poorly characterized pharmacokinetics. There are two binding sites per ACE (high affinity "C", lower affinity "N") that have sub-nanomolar affinities and dissociation rates of hours. Most inhibito...

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Detalles Bibliográficos
Main Authors: Levitt, David G, Schoemaker, Rik C
Formato: Artigo
Idioma:Inglês
Publicado: BioMed Central 2006
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC1373666/
https://ncbi.nlm.nih.gov/pubmed/16398929
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/1472-6904-6-1
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