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Growth inhibition and apoptosis induced by daunomycin-conjugated triplex-forming oligonucleotides targeting the c-myc gene in prostate cancer cells

Covalent attachment of intercalating agents to triplex-forming oligonucleotides (TFOs) is a promising strategy to enhance triplex stability and biological activity. We have explored the possibility to use the anticancer drug daunomycin as triplex stabilizing agent. Daunomycin-conjugated TFOs (dauno-...

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Библиографические подробности
Главные авторы: Napoli, Sara, Negri, Umberto, Arcamone, Federico, Capobianco, Massimo L., Carbone, Giuseppina M., Catapano, Carlo V.
Формат: Artigo
Язык:Inglês
Опубликовано: Oxford University Press 2006
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC1356532/
https://ncbi.nlm.nih.gov/pubmed/16449206
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkj473
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