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Phosphorylation of Ribavirin and Viramidine by Adenosine Kinase and Cytosolic 5′-Nucleotidase II: Implications for Ribavirin Metabolism in Erythrocytes

Many nucleoside analog drugs, such as ribavirin and viramidine, are activated or metabolized in vivo through 5′-phosphorylation. In this report, we determined the steady-state kinetic parameters for 5′-monophosphorylation of ribavirin and viramidine by adenosine kinase. The apparent K(m) for ribavir...

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Détails bibliographiques
Auteurs principaux: Wu, Jim Zhen, Larson, Gary, Walker, Heli, Shim, Jae Hoon, Hong, Zhi
Format: Artigo
Langue:Inglês
Publié: American Society for Microbiology 2005
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC1140532/
https://ncbi.nlm.nih.gov/pubmed/15917509
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.49.6.2164-2171.2005
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