Загрузка...

Antiretroviral Efficacy and Pharmacokinetics of Oral Bis(isopropyloxycarbonyloxymethyl)9-(2-Phosphonylmethoxypropyl)adenine in Mice

To overcome the low oral bioavailability of the highly potent and selective antiretroviral agent (R)-9-(2-phosphonylmethoxypropyl)adenine (PMPA), a new lipophilic ester derivative, i.e., the bis(isopropyloxycarbonyloxymethyl)-ester [bis(POC)-PMPA], was prepared. The usefulness of bis(POC)-PMPA as an...

Полное описание

Сохранить в:
Библиографические подробности
Главные авторы: Naesens, Lieve, Bischofberger, Norbert, Augustijns, Patrick, Annaert, Pieter, Van den Mooter, Guy, Arimilli, Murty N., Kim, Choung U., De Clercq, Erik
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Microbiology 1998
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC105646/
https://ncbi.nlm.nih.gov/pubmed/9660984
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!