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Phosphorus containing analogues of SAHA as inhibitors of HDACs

Histone deacetylases (HDACs) are a family of enzymes responsible for regulating DNA transcription by modulating its binding to histone proteins. HDACs are overexpressed in several types of cancers and are recognised as drug targets. Vorinostat, or suberanilohydroxamic acid (SAHA), is an histone deac...

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Autores principales: Michael D. Pun, Hsin-Hua Wu, Feyisola P. Olatunji, Britany N. Kesic, John W. Peters, Clifford E. Berkman
Formato: Artigo
Lenguaje:Inglês
Publicado: Taylor & Francis Group 2022-12-01
Colección:Journal of Enzyme Inhibition and Medicinal Chemistry
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Acceso en línea:https://www.tandfonline.com/doi/10.1080/14756366.2022.2063281
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