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A Series of Novel 1-<i>H</i>-isoindole-1,3(2<i>H</i>)-dione Derivatives as Acetylcholinesterase and Butyrylcholinesterase Inhibitors: In Silico, Synthesis and In Vitro Studies

The derivatives of isoindoline-1,3-dione are interesting due to their biological activities, such as anti-inflammatory and antibacterial effects. Several series have been designed and evaluated for Alzheimer’s therapy candidates. They showed promising activity. In this work, six new derivatives were...

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Autors principals: Edward Krzyżak, Aleksandra Marciniak, Dominika Szkatuła, Klaudia A. Jankowska, Natalia Dobies, Aleksandra Kotynia
Format: Artigo
Idioma:Inglês
Publicat: MDPI AG 2024-07-01
Col·lecció:Molecules
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Accés en línia:https://www.mdpi.com/1420-3049/29/15/3528
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