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Design, Synthesis, and Antibacterial Screening of Some Novel Heteroaryl-Based Ciprofloxacin Derivatives as DNA Gyrase and Topoisomerase IV Inhibitors

A novel series of ciprofloxacin hybrids comprising various heterocycle derivatives has been synthesized and structurally elucidated using <sup>1</sup>H NMR, <sup>13</sup>C NMR, and elementary analyses. Using ciprofloxacin as a reference, compounds <b>1–21</b> were screened in vitro against Gram-posi...

Повний опис

Збережено в:
Бібліографічні деталі
Автори: Lamya H. Al-Wahaibi, Amer A. Amer, Adel A. Marzouk, Hesham A. M. Gomaa, Bahaa G. M. Youssif, Antar A. Abdelhamid
Формат: Artigo
Мова:Inglês
Опубліковано: MDPI AG 2021-04-01
Серія:Pharmaceuticals
Предмети:
Онлайн доступ:https://www.mdpi.com/1424-8247/14/5/399
Теги: Додати тег
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