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Design, synthesis, and anti-Staphylococcus aureus evaluation of quinazolinone-based FabH inhibitors

Multidrug-resistant Staphylococcus aureus sparks global crisis and novel fatty acid synthesis enzyme FabH inhibitors could overcome resistance. Through rational design, we developed a series of quinazolinone-benzodioxin FabH inhibitors. The results showed that some of the newly synthesized compounds...

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Библиографические подробности
Главные авторы: Zi-Miao Wu, Meng-Jia Xu, Xiao-Meng Guo, Jian-Ke Ma, Xiu-Ling Gu, Li Cheng, Juan Sun
Формат: Artigo
Язык:Inglês
Опубликовано: Elsevier 2025-11-01
Серии:Results in Chemistry
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Online-ссылка:http://www.sciencedirect.com/science/article/pii/S2211715625008483
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