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Design, Synthesis, and Docking Study of Acyl Thiourea Derivatives as Possible Histone Deacetylase Inhibitors with a Novel Zinc Binding Group

Histone deacetylase inhibitors with zinc binding groups often exhibit drawbacks like non-selectivity or toxic effects. Thus, there are continuous efforts to modify the currently available inhibitors or to discover new derivatives to overcome these problems. One approach is to synthesize new compound...

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Збережено в:
Бібліографічні деталі
Автори: Duraid H. Al-Amily, Mohammed Hassan Mohammed
Формат: Artigo
Мова:Inglês
Опубліковано: MDPI AG 2019-10-01
Серія:Scientia Pharmaceutica
Предмети:
Онлайн доступ:https://www.mdpi.com/2218-0532/87/4/28
Теги: Додати тег
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