In Vitro Enzymatic and Kinetic Studies, and In Silico Drug-Receptor Interactions, and Drug-Like Profiling of the 5-Styrylbenzamide Derivatives as Potential Cholinesterase and β-Secretase Inhibitors with Antioxidant Properties

The 5-(styryl)anthranilamides were transformed into the corresponding 5-styryl-2-(<i>p</i>-tolylsulfonamido)benzamide derivatives. These 5-styrylbenzamide derivatives were evaluated through enzymatic assays in vitro for their capability to inhibit acetylcholinesterase (AChE), butyrylcholinesterase (...

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Bibliografski detalji

Glavni autori:	Malose J. Mphahlele, Emmanuel N. Agbo, Garland K. More, Samantha Gildenhuys
Format:	Artigo
Jezik:	Inglês
Izdano:	MDPI AG 2021-04-01
Serija:	Antioxidants
Teme:	5-styrylbenzamides cholinesterase β-secretase antioxidant metal chelating drug-receptor interactions
Online pristup:	https://www.mdpi.com/2076-3921/10/5/647
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