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Non-Canonical, Strongly Selective Protein Disulfide Isomerases as Anticancer Therapeutic Targets

Protein Disulfide Isomerases (PDIs) are emerging targets in anticancer therapy, with several PDI inhibitors demonstrating anticancer efficacy in preclinical models. Research has largely focused on “canonical” PDIs, such as PDIA1, which contain CXXC active site motifs where C represents Cysteine. Can...

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Váldodahkkit: Mary E. Law, Zaafir M. Dulloo, Brian Hardy, Ania Kelegama, Reagan Clark, Mariana Rivas Montbrun, Gabriella Antmann, Srihith Nooka, Ronald K. Castellano, Brian K. Law
Materiálatiipa: Artigo
Giella:Inglês
Almmustuhtton: MDPI AG 2025-08-01
Ráidu:Biomolecules
Fáttát:
Liŋkkat:https://www.mdpi.com/2218-273X/15/8/1146
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