Recent Advances in the Design, Synthesis, and Biological Evaluation of Selective DYRK1A Inhibitors: A New Avenue for a Disease Modifying Treatment of Alzheimer’s?

Por Smith, Breland, Medda, Federico, Gokhale, Vijay, Dunckley, Travis, Hulme, Christopher
Publicado em 2012

Synthesis and Biological Activity of 2-Aminothiazoles as Novel Inhibitors of PGE(2) Production in Cells

Por Smith, Breland, Chang, Hui-Hua, Medda, Federico, Gokhale, Vijay, Dietrich, Justin, Davis, Angela, Meuillet, Emmanuelle J., Hulme, Christopher
Publicado em 2012

Synthesis and biological activity of aminophthalazines and aminopyridazines as novel inhibitors of PGE(2) production in cells

Por Medda, Federico, Sells, Earlphia, Chang, Hui-Hua, Dietrich, Justin, Chappeta, Shashi, Smith, Breland, Gokhale, Vijay, Meuillet, Emmanuelle J., Hulme, Christopher
Publicado em 2012

Dyrk1 inhibition improves Alzheimer's disease‐like pathology

Por Branca, Caterina, Shaw, Darren M., Belfiore, Ramona, Gokhale, Vijay, Shaw, Arthur Y., Foley, Christopher, Smith, Breland, Hulme, Christopher, Dunckley, Travis, Meechoovet, Bessie, Caccamo, Antonella, Oddo, Salvatore
Publicado no Aging Cell (2017)