Impact of WIN site inhibitor on the WDR5 interactome

per Guarnaccia, Alissa D., Rose, Kristie L., Wang, Jing, Zhao, Bin, Popay, Tessa M., Wang, Christina E., Guerrazzi, Kiana, Hill, Salisha, Woodley, Chase M., Hansen, Tyler J., Lorey, Shelly L., Shaw, J. Grace, Payne, William G., Weissmiller, April M., Olejniczak, Edward T., Fesik, Stephen W., Liu, Qi, Tansey, William P.
Publicat a Cell Rep (2021)

Discovery and Structure-Based Optimization of Potent and Selective WDR5 Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core

per Tian, Jianhua, Teuscher, Kevin B., Aho, Erin R., Alvarado, Joseph R., Mills, Jonathan J., Meyers, Kenneth M., Gogliotti, Rocco D., Han, Changho, Macdonald, Jonathan D., Sai, Jiqing, Shaw, J. Grace, Sensintaffar, John L., Zhao, Bin, Rietz, Tyson A., Thomas, Lance R., Payne, William G., Moore, William J., Stott, Gordon M., Kondo, Jumpei, Inoue, Masahiro, Coffey, Robert J., Tansey, William P., Stauffer, Shaun R., Lee, Taekyu, Fesik, Stephen W.
Publicat a J Med Chem (2020)