Discovery of JTZ-951: A HIF Prolyl Hydroxylase Inhibitor for the Treatment of Renal Anemia

Por Ogoshi, Yosuke, Matsui, Takuya, Mitani, Ikuo, Yokota, Masahiro, Terashita, Masakazu, Motoda, Dai, Ueyama, Kazuhito, Hotta, Takahiro, Ito, Takashi, Hase, Yasunori, Fukui, Kenji, Deai, Katsuya, Yoshiuchi, Hiromi, Ito, Soichiro, Abe, Hiroyuki
Publicado no ACS Med Chem Lett (2017)

SAR Exploration Guided by LE and Fsp(3): Discovery of a Selective and Orally Efficacious RORγ Inhibitor

Por Hirata, Kazuyuki, Kotoku, Masayuki, Seki, Noriyoshi, Maeba, Takaki, Maeda, Katsuya, Hirashima, Shintaro, Sakai, Takayuki, Obika, Shingo, Hori, Akimi, Hase, Yasunori, Yamaguchi, Takayuki, Katsuda, Yoshiaki, Hata, Takahiro, Miyagawa, Naoki, Arita, Kojo, Nomura, Yukihiro, Asahina, Kota, Aratsu, Yusuke, Kamada, Masafumi, Adachi, Tsuyoshi, Noguchi, Masato, Doi, Satoki, Crowe, Paul, Bradley, Erin, Steensma, Ruo, Tao, Haiyan, Fenn, Morgan, Babine, Robert, Li, Xiaolin, Thacher, Scott, Hashimoto, Hiromasa, Shiozaki, Makoto
Publicado no ACS Med Chem Lett (2015)