Loading...
Efficient Synthesis of 1,4-Thiazepanones and 1,4-Thiazepanes as 3D Fragments for Screening Libraries
1,4-Thiazepanes and 1,4-thiazepanones represent seven-membered ring systems with highly 3D character and are currently underrepresented in fragment screening libraries. A nuclear magnetic resonance (NMR) fragment screen identified 1,4-acylthiazepanes as new BET (bromodomain and extraterminal domain)...
Na minha lista:
| Udgivet i: | Org Lett |
|---|---|
| Main Authors: | , , , , , |
| Format: | Artigo |
| Sprog: | Inglês |
| Udgivet: |
2020
|
| Fag: | |
| Online adgang: | https://ncbi.nlm.nih.gov/pmc/articles/PMC8324318/ https://ncbi.nlm.nih.gov/pubmed/32347732 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.orglett.0c01230 |
| Tags: |
Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!
|