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Synthesis and Cytotoxicity Evaluation of Spirocyclic Bromotyrosine Clavatadine C Analogs

Marine-originated spirocyclic bromotyrosines are considered as promising scaffolds for new anticancer drugs. In a continuation of our research to develop potent and more selective anticancer compounds, we synthesized a library of 32 spirocyclic clavatadine analogs by replacing the agmatine, i.e., 4-...

詳細記述

保存先:
書誌詳細
出版年:Mar Drugs
主要な著者: Patel, Piyush A., Bruun, Tanja, Ilina, Polina, Mäkkylä, Heidi, Lempinen, Antti, Yli-Kauhaluoma, Jari, Tammela, Päivi, Kiuru, Paula S.
フォーマット: Artigo
言語:Inglês
出版事項: MDPI 2021
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC8305101/
https://ncbi.nlm.nih.gov/pubmed/34356825
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md19070400
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