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A Novel Triphenylphosphonium Carrier to Target Mitochondria without Uncoupling Oxidative Phosphorylation

Mitochondrial dysfunction is an underlying pathology in numerous diseases. Delivery of diagnostic and therapeutic cargo directly into mitochondria is a powerful approach to study and treat these diseases. The triphenylphosphonium (TPP(+)) moiety is the most widely used mitochondriotropic carrier. Ho...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Kulkarni, Chaitanya A., Fink, Brian D., Gibbs, Bettine E., Chheda, Pratik R., Wu, Meng, Sivitz, William I., Kerns, Robert J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2021
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8293692/
https://ncbi.nlm.nih.gov/pubmed/33395531
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.0c01671
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