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Inhibition of Nav1.7 channel by a novel blocker QLS-81 for alleviation of neuropathic pain

Voltage-gated sodium channel Nav1.7 robustly expressed in peripheral nociceptive neurons has been considered as a therapeutic target for chronic pain, but there is no selective Nav1.7 inhibitor available for therapy of chronic pain. Ralfinamide has shown anti-nociceptive activity in animal models of...

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Bibliografski detalji
Izdano u:Acta Pharmacol Sin
Glavni autori: Niu, He-ling, Liu, Ya-ni, Xue, Deng-qi, Dong, Li-ying, Liu, Hui-jie, Wang, Jing, Zheng, Yi-lin, Zou, An-ruo, Shao, Li-ming, Wang, KeWei
Format: Artigo
Jezik:Inglês
Izdano: Springer Singapore 2021
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC8285378/
https://ncbi.nlm.nih.gov/pubmed/34103689
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41401-021-00682-9
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