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Toward New Transmission-Blocking Combination Therapies: Pharmacokinetics of 10-Amino-Artemisinins and 11-Aza-Artemisinin and Comparison with Dihydroartemisinin and Artemether

As artemisinin combination therapies (ACTs) are compromised by resistance, we are evaluating triple combination therapies (TACTs) comprising an amino-artemisinin, a redox drug, and a third drug with a different mode of action. Thus, here we briefly review efficacy data on artemisone, artemiside, oth...

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Detalhes bibliográficos
Publicado no:Antimicrob Agents Chemother
Main Authors: Watson, Daniel J., Laing, Lizahn, Gibhard, Liezl, Wong, Ho Ning, Haynes, Richard K., Wiesner, Lubbe
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8284440/
https://ncbi.nlm.nih.gov/pubmed/34097488
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00990-21
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