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Synthesis and biological evaluation of 5-aminoethyl benzophenanthridone derivatives as DNA topoisomerase IB inhibitors

DNA topoisomerase IB (TOP1) regulates DNA topological structure in many cellular metabolic processes and is a validated target for development of antitumor agents. Our previous study revealed that the benzophenanthridone scaffold is a novel chemotype for the discovery of TOP1 inhibitors. In this wor...

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Publicat a:Eur J Med Chem
Autors principals: Tang, Wen-Lin, Zhang, Yu, Hu, De-Xuan, Yang, Hui, Yu, Qian, Chen, Jian-Wen, Agama, Keli, Pommier, Yves, An, Lin-Kun
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8274952/
https://ncbi.nlm.nih.gov/pubmed/31176097
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2019.05.074
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