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Acridones are Highly Potent Inhibitors of Toxoplasma gondii Tachyzoites

Acridone derivatives, which have been shown to have in vitro and in vivo activity against Plasmodium spp, inhibit Toxoplasma gondii proliferation at picomolar concentrations. Using enzymatic assays, we show that acridones inhibit both T. gondii cytochrome bc(1) and dihydroorotate dehydrogenase and i...

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Vydáno v:ACS Infect Dis
Hlavní autoři: Alday, P. Holland, McConnell, Erin V., Boitz Zarella, Jan M., Dodean, Rozalia A., Kancharla, Papireddy, Kelly, Jane X., Doggett, J. Stone
Médium: Artigo
Jazyk:Inglês
Vydáno: 2021
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC8273083/
https://ncbi.nlm.nih.gov/pubmed/33723998
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.1c00016
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