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The Research Progress of Direct KRAS G12C Mutation Inhibitors

Abstract: KRAS mutations have long been considered undruggable. However, a series of direct KRAS mutation inhibitors have been developed since the switch II pocket was discovered recently. This review will summarize progress in the development of direct KRAS G12C mutation inhibitors, current relevan...

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Publicat a:Pathol Oncol Res
Autors principals: Yang, Ai, Li, Min, Fang, Mingzhi
Format: Artigo
Idioma:Inglês
Publicat: Frontiers Media S.A. 2021
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8262225/
https://ncbi.nlm.nih.gov/pubmed/34257597
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/pore.2021.631095
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