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New quinoline-triazole conjugates: Synthesis, and antiviral properties against SARS-CoV-2

At present therapeutic options for severe acute respiratory syndrome coronavirus-2 (SARS-CoV-2) are very limited. We designed and synthesized three sets of small molecules using quinoline scaffolds. A series of quinoline conjugates (10a-l, 11a-c, and 12a-e) by incorporating 1,2,3-triazole were synth...

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Bibliografske podrobnosti
izdano v:Bioorg Chem
Main Authors: Seliem, Israa A., Panda, Siva S., Girgis, Adel S., Moatasim, Yassmin, Kandeil, Ahmed, Mostafa, Ahmed, Ali, Mohamed A., Nossier, Eman S., Rasslan, Fatma, Srour, Aladdin M., Sakhuja, Rajeev, Ibrahim, Tarek S., Abdel-samii, Zakaria K.M., Al-Mahmoudy, Amany M.M.
Format: Artigo
Jezik:Inglês
Izdano: Elsevier Inc. 2021
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC8219945/
https://ncbi.nlm.nih.gov/pubmed/34214752
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bioorg.2021.105117
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