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Cancer Selective Target Degradation by Folate-Caged PROTACs

PROTACs (proteolysis targeting chimeras) are an emerging class of promising therapeutic modalities that degrade intracellular protein targets by hijacking the cellular ubiquitin–proteasome system. However, potential toxicity of PROTACs in normal cells due to the off-tissue on-target degradation effe...

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Detalles Bibliográficos
Publicado en:J Am Chem Soc
Autores principales: Liu, Jing, Chen, He, Liu, Yi, Shen, Yudao, Meng, Fanye, Kaniskan, H. ϋmit, Jin, Jian, Wei, Wenyi
Formato: Artigo
Lenguaje:Inglês
Publicado: 2021
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC8219215/
https://ncbi.nlm.nih.gov/pubmed/33970635
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.1c00451
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