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Concise Chemoenzymatic Total Synthesis and Identification of Cellular Targets of Cepafungin I

The natural product cepafungin I was recently reported to be one of the most potent covalent inhibitors of the 20S proteasome core particle through a series of in vitro activity assays. Here, we report a short chemoenzymatic total synthesis of cepafungin I featuring the use of a regioselective enzym...

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Bibliographic Details
Published in:Cell Chem Biol
Main Authors: Amatuni, Alexander, Shuster, Anton, Adibekian, Alexander, Renata, Hans
Format: Artigo
Language:Inglês
Published: 2020
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC8201661/
https://ncbi.nlm.nih.gov/pubmed/32763140
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2020.07.012
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