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Using Chemical Structure Information to Develop Predictive Models for In Vitro Toxicokinetic Parameters to Inform High-throughput Risk-assessment

The toxicokinetic (TK) parameters fraction of the chemical unbound to plasma proteins and metabolic clearance are critical for relating exposure and internal dose when building in vitro-based risk assessment models. However, experimental toxicokinetic studies have only been carried out on limited ch...

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Podrobná bibliografie
Vydáno v:Comput Toxicol
Hlavní autoři: Pradeep, Prachi, Patlewicz, Grace, Pearce, Robert, Wambaugh, John, Wetmore, Barbara, Judson, Richard
Médium: Artigo
Jazyk:Inglês
Vydáno: 2020
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC8193769/
https://ncbi.nlm.nih.gov/pubmed/34124416
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.comtox.2020.100136
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