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Inhibitors of thiol-mediated uptake

Ellman's reagent has caused substantial confusion and concern as a probe for thiol-mediated uptake because it is the only established inhibitor available but works neither efficiently nor reliably. Here we use fluorescent cyclic oligochalcogenides that enter cells by thiol-mediated uptake to sy...

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Publicat a:Chem Sci
Autors principals: Cheng, Yangyang, Pham, Anh-Tuan, Kato, Takehiro, Lim, Bumhee, Moreau, Dimitri, López-Andarias, Javier, Zong, Lili, Sakai, Naomi, Matile, Stefan
Format: Artigo
Idioma:Inglês
Publicat: The Royal Society of Chemistry 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8179002/
https://ncbi.nlm.nih.gov/pubmed/34163793
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0sc05447j
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