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Elementary mechanisms of calmodulin regulation of Na(V)1.5 producing divergent arrhythmogenic phenotypes

In cardiomyocytes, Na(V)1.5 channels mediate initiation and fast propagation of action potentials. The Ca(2+)-binding protein calmodulin (CaM) serves as a de facto subunit of Na(V)1.5. Genetic studies and atomic structures suggest that this interaction is pathophysiologically critical, as human muta...

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Detalhes bibliográficos
Publicado no:Proc Natl Acad Sci U S A
Main Authors: Kang, Po Wei, Chakouri, Nourdine, Diaz, Johanna, Tomaselli, Gordon F., Yue, David T., Ben-Johny, Manu
Formato: Artigo
Idioma:Inglês
Publicado em: National Academy of Sciences 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8166197/
https://ncbi.nlm.nih.gov/pubmed/34021086
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.2025085118
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