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Substance P Serves as a Balanced Agonist for MRGPRX2 and a Single Tyrosine Residue Is Required for β-Arrestin Recruitment and Receptor Internalization

The neuropeptide substance P (SP) mediates neurogenic inflammation and pain and contributes to atopic dermatitis in mice through the activation of mast cells (MCs) via Mas-related G protein-coupled receptor (GPCR)-B2 (MrgprB2, human ortholog MRGPRX2). In addition to G proteins, certain MRGPRX2 agoni...

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Dades bibliogràfiques
Publicat a:Int J Mol Sci
Autors principals: Chompunud Na Ayudhya, Chalatip, Amponnawarat, Aetas, Ali, Hydar
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8158387/
https://ncbi.nlm.nih.gov/pubmed/34070125
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms22105318
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