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Physicochemical properties and Mycobacterium tuberculosis transporters: keys to efficacious antitubercular drugs?

Securing novel, safe, and effective medicines to treat Mycobacterium tuberculosis remains an elusive goal, particularly influenced by the largely impervious Mtb envelope that limits exposure and thus efficacy of inhibitors at their cellular and periplasmic targets. The impact of physicochemical prop...

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Библиографические подробности
Опубликовано в: :RSC Med Chem
Главные авторы: Fullam, Elizabeth, Young, Robert J.
Формат: Artigo
Язык:Inglês
Опубликовано: RSC 2020
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC8130550/
https://ncbi.nlm.nih.gov/pubmed/34041481
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0md00265h
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