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Synthetic Tuning of Domain Stoichiometry in Nanobody–Enzyme Megamolecules

This paper presents a method to synthetically tune atomically precise megamolecule nanobody–enzyme conjugates for prodrug cancer therapy. Previous efforts to create heterobifunctional protein conjugates suffered from heterogeneity in domain stoichiometry, which in part led to the failure of antibody...

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Dades bibliogràfiques
Publicat a:Bioconjug Chem
Autors principals: Metcalf, Kevin J., Kimmel, Blaise R., Sykora, Daniel J., Modica, Justin A., Parker, Kelly A., Berens, Eric, Dai, Raymond, Dravid, Vinayak P., Werb, Zena, Mrksich, Milan
Format: Artigo
Idioma:Inglês
Publicat: 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8109025/
https://ncbi.nlm.nih.gov/pubmed/33301672
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.bioconjchem.0c00578
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