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Mechanism of covalent binding of ibrutinib to Bruton's tyrosine kinase revealed by QM/MM calculations

Ibrutinib is the first covalent inhibitor of Bruton's tyrosine kinase (BTK) to be used in the treatment of B-cell cancers. Understanding the mechanism of covalent inhibition will aid in the design of safer and more selective covalent inhibitors that target BTK. The mechanism of covalent inhibit...

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Bibliografische gegevens
Gepubliceerd in:Chem Sci
Hoofdauteurs: Voice, Angus T., Tresadern, Gary, Twidale, Rebecca M., van Vlijmen, Herman, Mulholland, Adrian J.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: The Royal Society of Chemistry 2021
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8097726/
https://ncbi.nlm.nih.gov/pubmed/33995994
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0sc06122k
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