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The impact of cytochrome P450 3A genetic polymorphisms on tacrolimus pharmacokinetics in ulcerative colitis patients

Tacrolimus (Tac) is an effective remission inducer of refractory ulcerative colitis (UC). Gene polymorphisms result in interindividual variability in Tac pharmacokinetics. In this study, we aimed to examine the relationships between gene polymorphisms and the metabolism, pharmacokinetics, and therap...

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書目詳細資料
發表在:PLoS One
Main Authors: Furuse, Maizumi, Hosomi, Shuhei, Nishida, Yu, Itani, Shigehiro, Nadatani, Yuji, Fukunaga, Shusei, Otani, Koji, Tanaka, Fumio, Nagami, Yasuaki, Taira, Koichi, Kamata, Noriko, Watanabe, Toshio, Watanabe, Kenji, Fujiwara, Yasuhiro
格式: Artigo
語言:Inglês
出版: Public Library of Science 2021
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC8062093/
https://ncbi.nlm.nih.gov/pubmed/33886687
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0250597
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