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Comparative Activity and Off-Target Effects in Cells of the CHK1 Inhibitors MK-8776, SRA737, and LY2606368

[Image: see text] DNA damage activates the checkpoint protein CHK1 to arrest cell cycle progression, providing time for repair and recovery. Consequently, inhibitors of CHK1 (CHK1i) enhance damage-induced cell death. Additionally, CHK1i elicits single agent cytotoxicity in some cell lines. We compar...

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Bibliografske podrobnosti
izdano v:ACS Pharmacol Transl Sci
Main Authors: Ditano, Jennifer P., Eastman, Alan
Format: Artigo
Jezik:Inglês
Izdano: American Chemical Society 2021
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC8033610/
https://ncbi.nlm.nih.gov/pubmed/33860197
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsptsci.0c00201
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