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NHERF1/EBP50 as a Target for Modulation of MRP Function in HepG2 Cells

As increased expression and activities of efflux transporters (ETs) often cause drug resistance in cancers, we tried modulating ET activity in cancer cells, using scaffold proteins such as ezrin/radixin/moesin (ERM) proteins, and Na(+)/H(+) exchanger regulatory factor-1 (NHERF1)/ERM-binding phosphop...

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Publicat a:Pharmaceuticals (Basel)
Autors principals: Kawase, Atsushi, Hirosoko, Miho, Sugihara, Yuka, Koyama, Yunosuke, Fukae, Ayaka, Shimada, Hiroaki, Iwaki, Masahiro
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8002045/
https://ncbi.nlm.nih.gov/pubmed/33800412
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph14030239
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