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NHERF1/EBP50 as a Target for Modulation of MRP Function in HepG2 Cells

As increased expression and activities of efflux transporters (ETs) often cause drug resistance in cancers, we tried modulating ET activity in cancer cells, using scaffold proteins such as ezrin/radixin/moesin (ERM) proteins, and Na(+)/H(+) exchanger regulatory factor-1 (NHERF1)/ERM-binding phosphop...

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Detalhes bibliográficos
Publicado no:Pharmaceuticals (Basel)
Main Authors: Kawase, Atsushi, Hirosoko, Miho, Sugihara, Yuka, Koyama, Yunosuke, Fukae, Ayaka, Shimada, Hiroaki, Iwaki, Masahiro
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8002045/
https://ncbi.nlm.nih.gov/pubmed/33800412
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph14030239
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