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Synthesis of Two Methotrexate Prodrugs for Optimizing Drug Loading into Liposomes

Methotrexate (MTX), a compound originally used as an anticancer drug, has also found applications in a broad variety of autoimmune disorders thanks to its anti-inflammation and immunomodulatory functions. The broad application of MTX is anyway limited by its poor solubility in biological fluids, its...

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Detalhes bibliográficos
Publicado no:Pharmaceutics
Main Authors: Di Francesco, Valentina, Di Francesco, Martina, Decuzzi, Paolo, Palomba, Roberto, Ferreira, Miguel
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7998143/
https://ncbi.nlm.nih.gov/pubmed/33806703
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics13030332
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