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Inhibition of RAF dimers: it takes two to tango

The RAS-regulated RAF–MEK1/2–ERK1/2 pathway promotes cell proliferation and survival and RAS and BRAF proteins are commonly mutated in cancer. This has fuelled the development of small molecule kinase inhibitors including ATP-competitive RAF inhibitors. Type I and type I½ ATP-competitive RAF inhibit...

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Pubblicato in:Biochem Soc Trans
Autori principali: Cook, Frazer A., Cook, Simon J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Portland Press Ltd. 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7924995/
https://ncbi.nlm.nih.gov/pubmed/33367512
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BST20200485
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