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Discovery of sultam-containing small-molecule disruptors of the huntingtin—calmodulin protein—protein interaction

The aberrant protein—protein interaction between calmodulin and mutant huntingtin protein in Huntington’s disease patients has been found to contribute to Huntington’s disease progression. A high-throughput screen for small molecules capable of disrupting this interaction revealed a sultam series as...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Med Chem Res
Päätekijät: Klus, Nicholas J., Kapadia, Khushboo, McDonald, Peter, Roy, Anuradha, Frankowski, Kevin J., Muma, Nancy A., Aubé, Jeffrey
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2020
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC7906539/
https://ncbi.nlm.nih.gov/pubmed/33642842
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00044-020-02583-8
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