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WIDOCK: a reactive docking protocol for virtual screening of covalent inhibitors

Here we present WIDOCK, a virtual screening protocol that supports the selection of diverse electrophiles as covalent inhibitors by incorporating ligand reactivity towards cysteine residues into AutoDock4. WIDOCK applies the reactive docking method (Backus et al. in Nature 534:570–574, 2016) and ext...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:J Comput Aided Mol Des
Egile Nagusiak: Scarpino, Andrea, Petri, László, Knez, Damijan, Imre, Tímea, Ábrányi-Balogh, Péter, Ferenczy, György G., Gobec, Stanislav, Keserű, György M.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Springer International Publishing 2021
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7904743/
https://ncbi.nlm.nih.gov/pubmed/33458809
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-020-00371-5
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