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G-quadruplex binding properties of a potent PARP-1 inhibitor derived from 7-azaindole-1-carboxamide

Poly ADP-ribose polymerases (PARP) are key proteins involved in DNA repair, maintenance as well as regulation of programmed cell death. For this reason they are important therapeutic targets for cancer treatment. Recent studies have revealed a close interplay between PARP1 recruitment and G-quadrupl...

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Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Dallavalle, Sabrina, Musso, Loana, Artali, Roberto, Aviñó, Anna, Scaglioni, Leonardo, Eritja, Ramon, Gargallo, Raimundo, Mazzini, Stefania
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7887208/
https://ncbi.nlm.nih.gov/pubmed/33594142
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-021-83474-9
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